Items where Author is "Radi, Marco"

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Number of items: 10.

Article

Castagnolo, Daniele, Scalacci, Nicolò, Pelloja, Chiara and Radi, Marco (2016) Microwave-assisted domino reactions of propargylamines with isothiocyanates: selective synthesis of 2-aminothiazoles and 2-amino-4-methylenethiazolines. Synlett, 27 (12). pp. 1883-1887. ISSN 0936-5214

Vincetti, Paolo, Brianza, Anna, Scalacci, Nicolò, Costantino, Gabriele, Castagnolo, Daniele and Radi, Marco (2016) A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides. Tetrahedron Letters, 57 (13). pp. 1464-1467. ISSN 0040-4039

Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolò, Kissova, Miroslava, Armijos-Rivera, Jorge, Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele and Radi, Marco (2016) A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes. MedChemComm, 7 (3). pp. 484-494. ISSN 2040-2503

Magri, Andrea, Reilly, Roisin, Scalacci, Nicolò, Radi, Marco, Hunter, Michael, Ripoll, Manon, Patel, Arvind H. and Castagnolo, Daniele (2015) Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents. Bioorganic & Medicinal Chemistry Letters, 25 (22). pp. 5372-5376. ISSN 0960-894X

Vincetti, Paolo, Caporuscio, Fabiana, Kaptein, Suzanne, Gioiello, Antimo, Mancino, Valentina, Suzuki, Youichi, Yamamoto, Naoki, Crespan, Emmanuele, Lossani, Andrea, Maga, Giovanni, Rastelli, Giulio, Castagnolo, Daniele, Neyts, Johan, Leyssen, Pieter, Costantino, Gabriele and Radi, Marco (2015) Discovery of Multitarget Antivirals Acting on Both the Dengue Virus NS5-NS3 Interaction and the Host Src/Fyn Kinases. Journal of Medicinal Chemistry, 58 (12). pp. 4964-4975. ISSN 0022-2623

Radi, Marco, Pagano, Mafalda, Franchi, Luigi, Castagnolo, Daniele, Schenone, Silvia, Casaluce, Gianni, Zamperini, Claudio, Dreassi, Elena, Maga, Giovanni, Samuele, Alberta, Gonzalo, Encarna, Clotet, Bonaventura, Esté, José and Botta, Maurizio (2012) Synthesis, biological activity, and ADME properties of novel S-DABOs/N-DABOs as HIV reverse transcriptase inhibitors. ChemMedChem, 7 (5). pp. 883-896. ISSN 1860-7179

Schenone, Silvia, Brullo, Chiara, Musumeci, Francesca, Radi, Marco and Castagnolo, Daniele (2011) Src Kinase Inhibitors: An update on patented compounds. Current Medicinal Chemistry, 18 (33). pp. 5061-5078. ISSN 0929-8673

Radi, Marco, Bernardo, Vincenzo, Bechi, Beatrice, Castagnolo, Daniele, Pagano, Mafalda and Botta, Maurizio (2009) Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles. Tetrahedron Letters, 50 (47). pp. 6572-6575. ISSN 0040-4039

Castagnolo, Daniele, Manetti, Fabrizio, Radi, Marco, Bechi, Beatrice, Pagano, Mafalda, de Logu, Alessandro, Meleddu, Rita, Saddi, Manuela and Botta, Maurizio (2009) Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones. Bioorganic & Medicinal Chemistry, 17 (15). pp. 5716-5721. ISSN 0968-0896

Castagnolo, Daniele, de Logu, Alessandro, Radi, Marco, Bechi, Beatrice, Manetti, Fabrizio, Magnani, Matteo, Supino, Sibilla, Meleddu, Rita, Chisu, Lorenza and Botta, Maurizio (2008) Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis. Bioorganic & Medicinal Chemistry, 16 (18). pp. 8587-8591. ISSN 0968-0896

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