Items where Author is "Castagnolo, Daniele"

Article

Zhao, Fei, Masci, Domiziana, Ferla, Salvatore, Varricchio, Carmine, Brancale, Andrea, Colonna, Serena, Black, Gary, Turner, Nicholas J. and Castagnolo, Daniele (2020) Monoamine Oxidase (MAO-N) Biocatalyzed Synthesis of Indoles from Indolines Prepared via Photocatalytic Cyclization/Arylative Dearomatization. ACS Catalysis, 10 (11). pp. 6414-6421. ISSN 2155-5435

Lauder, Kate, Masci, Domiziana, Toscani, Anita, Al Mekdad, Aya, Black, Gary, Brown, Nicola, Turner, Nicholas J., Luisi, Renzo and Castagnolo, Daniele (2019) A facile and regioselective multicomponent synthesis of chiral aryl-1,2-mercaptoamines in water followed by monoamine oxidase (MAO-N) enzymatic resolution. Organic & Biomolecular Chemistry, 17 (40). pp. 8982-8986. ISSN 1477-0520

Toscani, Anita, Risi, Caterina, Black, Gary, Brown, Nicola, Shaaban, Ali, Turner, Nicholas J. and Castagnolo, Daniele (2018) Monoamine Oxidase (MAO-N) Whole Cell Biocatalyzed Aromatization of 1,2,5,6-Tetrahydropyridines into Pyridines. ACS Catalysis, 8 (9). pp. 8781-8787. ISSN 2155-5435

Castagnolo, Daniele, Bass, Rosemary, Jenkinson, Sarah, Wright, Jennifer, Smulders-Srinivasan, Tora and Marshall, Jamie (2017) Synthesis and biological evaluation of novel amidinourea and triazine congeners as inhibitors of MDA-MB-231 human breast cancer cell proliferation. ChemMedChem, 12 (4). pp. 288-291. ISSN 1860-7179

Scalacci, Nicolò, Brown, Alistair, Pavan, Fernando, Ribeiro, Camila, Manetti, Fabrizio, Bhakta, Sanjib, Maitra, Arundhati, Smith, Darren, Petricci, Elena and Castagnolo, Daniele (2017) Synthesis and SAR evaluation of novel thioridazine derivatives active against drug-resistant tuberculosis. European Journal of Medicinal Chemistry, 127. pp. 147-158. ISSN 0223-5234

Scalacci, Nicolò, Black, Gary, Mattedi, Giulio, Brown, Nicola, Turner, Nicholas J. and Castagnolo, Daniele (2017) Unveiling the Biocatalytic Aromatizing Activity of Monoamine Oxidases MAO-N and 6-HDNO: Development of Chemoenzymatic Cascades for the Synthesis of Pyrroles. ACS Catalysis, 7 (2). pp. 1295-1300. ISSN 2155-5435

Castagnolo, Daniele, Scalacci, Nicolò, Pelloja, Chiara and Radi, Marco (2016) Microwave-assisted domino reactions of propargylamines with isothiocyanates: selective synthesis of 2-aminothiazoles and 2-amino-4-methylenethiazolines. Synlett, 27 (12). pp. 1883-1887. ISSN 0936-5214

Vincetti, Paolo, Brianza, Anna, Scalacci, Nicolò, Costantino, Gabriele, Castagnolo, Daniele and Radi, Marco (2016) A microwave-assisted multicomponent protocol for the synthesis of benzofuran-2-carboxamides. Tetrahedron Letters, 57 (13). pp. 1464-1467. ISSN 0040-4039

Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolò, Kissova, Miroslava, Armijos-Rivera, Jorge, Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele and Radi, Marco (2016) A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes. MedChemComm, 7 (3). pp. 484-494. ISSN 2040-2503

Bhakta, Sanjib, Scalacci, Nicolò, Maitra, Arundhati, Brown, Alistair, Dasugari, Saiprasad, Evangelopoulos, Dimitrios, McHugh, Timothy, Mortazavi, Parisa, Twist, Alexander, Petricci, Elena, Manetti, Fabrizio and Castagnolo, Daniele (2016) Design and Synthesis of 1-((1,5-Bis(4-chlorophenyl)-2-methyl-1H-pyrrol-3-yl)methyl)-4-methylpiperazine (BM212) and N-Adamantan-2-yl-N′-((E)-3,7-dimethylocta-2,6-dienyl)ethane-1,2-diamine (SQ109) Pyrrole Hybrid Derivatives: Discovery of Potent Antitubercular Agents Effective against Multidrug-Resistant Mycobacteria. Journal of Medicinal Chemistry, 59 (6). pp. 2780-2793. ISSN 0022-2623

Magri, Andrea, Reilly, Roisin, Scalacci, Nicolò, Radi, Marco, Hunter, Michael, Ripoll, Manon, Patel, Arvind H. and Castagnolo, Daniele (2015) Rethinking the old antiviral drug moroxydine: Discovery of novel analogues as anti-hepatitis C virus (HCV) agents. Bioorganic & Medicinal Chemistry Letters, 25 (22). pp. 5372-5376. ISSN 0960-894X

Vincetti, Paolo, Caporuscio, Fabiana, Kaptein, Suzanne, Gioiello, Antimo, Mancino, Valentina, Suzuki, Youichi, Yamamoto, Naoki, Crespan, Emmanuele, Lossani, Andrea, Maga, Giovanni, Rastelli, Giulio, Castagnolo, Daniele, Neyts, Johan, Leyssen, Pieter, Costantino, Gabriele and Radi, Marco (2015) Discovery of Multitarget Antivirals Acting on Both the Dengue Virus NS5-NS3 Interaction and the Host Src/Fyn Kinases. Journal of Medicinal Chemistry, 58 (12). pp. 4964-4975. ISSN 0022-2623

Chachignon, Helene, Scalacci, Nicolò, Petricci, Elena and Castagnolo, Daniele (2015) Synthesis of 1,2,3-substituted pyrroles from propargylamines via a one-pot tandem enyne cross metathesis-cyclization reaction. Journal of Organic Chemistry, 80 (10). pp. 5287-5295. ISSN 0022-3263

Castagnolo, Daniele, Degennaro, Leonardo, Luisi, Renzo and Clayden, Jonathan (2015) Enantioselective carbolithiation of S-alkenyl-N-aryl thiocarbamates: kinetic and thermodynamic control. Organic and Biomolecular Chemistry, 13 (8). pp. 2330-2340. ISSN 1477-0520

Sanguinetti, Maurizio, Sanfilippo, Stefania, Castagnolo, Daniele, Sanglard, Dominique, Posteraro, Brunella, Donzellini, Giovanni and Botta, Maurizio (2013) Novel Macrocyclic Amidinoureas: Potent Non-Azole antifungals active against wild-type and resistant Candida species. ACS Medicinal Chemistry Letters, 4 (9). pp. 852-857. ISSN 1948-5875

Castagnolo, Daniele, Pagano, Mafalda, Bernardini, Martina and Botta, Maurizio (2012) Studies on the acylation of 4-(2-aminoethylthio)-7-nitrobenzofurazan: the role of bases in promoting the formation of fluorescent S-acyl derivatives through S–N Smiles rearrangement. Tetrahedron Letters, 53 (37). pp. 5008-5011. ISSN 0040-4039

Radi, Marco, Pagano, Mafalda, Franchi, Luigi, Castagnolo, Daniele, Schenone, Silvia, Casaluce, Gianni, Zamperini, Claudio, Dreassi, Elena, Maga, Giovanni, Samuele, Alberta, Gonzalo, Encarna, Clotet, Bonaventura, Esté, José and Botta, Maurizio (2012) Synthesis, biological activity, and ADME properties of novel S-DABOs/N-DABOs as HIV reverse transcriptase inhibitors. ChemMedChem, 7 (5). pp. 883-896. ISSN 1860-7179

Castagnolo, Daniele, Schenone, Silvia and Botta, Maurizio (2011) Guanylated Diamines, Triamines, and Polyamines: Chemistry and biological properties. Chemical Reviews, 111 (9). pp. 5247-5300. ISSN 0009-2665

Schenone, Silvia, Brullo, Chiara, Musumeci, Francesca, Radi, Marco and Castagnolo, Daniele (2011) Src Kinase Inhibitors: An update on patented compounds. Current Medicinal Chemistry, 18 (33). pp. 5061-5078. ISSN 0929-8673

Castagnolo, Daniele, Contemori, Lorenzo, Maccari, Giorgio, Avramova, Stanislava, Neri, Annalisa, Sgaragli, Gianpietro and Botta, Maurizio (2010) From taxuspine X to structurally simplified taxanes with remarkable P-Glycoprotein inhibitory activity. ACS Medicinal Chemistry Letters, 1 (8). pp. 416-421. ISSN 1948-5875

Castagnolo, Daniele and Botta, Maurizio (2010) Iron-catalyzed cross-coupling between 1-Bromoalkynes and Grignard-derived organocuprate reagents. European Journal of Organic Chemistry, 2010 (17). pp. 3224-3228. ISSN 1434-193X

Castagnolo, Daniele, Botta, Lorenzo and Botta, Maurizio (2009) Stereoselective protecting group free synthesis of d,l-gulose ethyl glycoside via multicomponent enyne cross metathesis—hetero Diels–Alder reaction. Carbohydrate Research, 344 (11). pp. 1285-1288. ISSN 0008-6215

Castagnolo, Daniele, Botta, Lorenzo and Botta, Maurizio (2009) Alkyne-enol ether cross-metathesis in the presence of CuSO4: Direct formation of 3-substituted crotonaldehydes in aqueous medium. The Journal of Organic Chemistry, 74 (8). pp. 3172-3174. ISSN 0022-3263

Botta, Maurizio, Castagnolo, Daniele, Pagano, Mafalda and Bernardini, Martina (2009) Domino alkylation-cyclization reaction of propargyl bromides with thioureas/thiopyrimidinones: A new facile synthesis of 2-aminothiazoles and 5H-thiazolo[3,2-a]pyrimidin-5-ones. Synlett, 2009 (13). pp. 2093-2096. ISSN 0936-5214

Castagnolo, Daniele, Raffi, Francesco, Giorgi, Gianluca and Botta, Maurizio (2009) Macrocyclization of Di-Boc-guanidino-alkylamines Related to Guazatine Components: Discovery and synthesis of innovative macrocyclic amidinoureas. European Journal of Organic Chemistry, 2009 (3). pp. 334-337. ISSN 1434-193X

Radi, Marco, Bernardo, Vincenzo, Bechi, Beatrice, Castagnolo, Daniele, Pagano, Mafalda and Botta, Maurizio (2009) Microwave-assisted organocatalytic multicomponent Knoevenagel/hetero Diels–Alder reaction for the synthesis of 2,3-dihydropyran[2,3-c]pyrazoles. Tetrahedron Letters, 50 (47). pp. 6572-6575. ISSN 0040-4039

Castagnolo, Daniele, Botta, Lorenzo and Botta, Maurizio (2009) One-pot multicomponent synthesis of 2,3-dihydropyrans: new access to furanose–pyranose 1,3-C–C-linked-disaccharides. Tetrahedron Letters, 50 (14). pp. 1526-1528. ISSN 0040-4039

Manetti, Fabrizio, Castagnolo, Daniele, Raffi, Francesco, Zizzari, Alessandra, Rajamäki, Suvi, D’Arezzo, Silvia, Visca, Paolo, Cona, Alessandra, Fracasso, Maria Enrica, Doria, Denise, Posteraro, Brunella, Sanguinetti, Maurizio, Fadda, Giovanni and Botta, Maurizio (2009) Synthesis of new linear guanidines and macrocyclic amidinourea derivatives endowed with high antifungal activity against Candida spp. and Aspergillus spp. Journal of Medicinal Chemistry, 52 (23). pp. 7376-7379. ISSN 0022-2623

Castagnolo, Daniele, Manetti, Fabrizio, Radi, Marco, Bechi, Beatrice, Pagano, Mafalda, de Logu, Alessandro, Meleddu, Rita, Saddi, Manuela and Botta, Maurizio (2009) Synthesis, biological evaluation, and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis: Part 2. Synthesis of rigid pyrazolones. Bioorganic & Medicinal Chemistry, 17 (15). pp. 5716-5721. ISSN 0968-0896

Castagnolo, Daniele, de Logu, Alessandro, Radi, Marco, Bechi, Beatrice, Manetti, Fabrizio, Magnani, Matteo, Supino, Sibilla, Meleddu, Rita, Chisu, Lorenza and Botta, Maurizio (2008) Synthesis, biological evaluation and SAR study of novel pyrazole analogues as inhibitors of Mycobacterium tuberculosis. Bioorganic & Medicinal Chemistry, 16 (18). pp. 8587-8591. ISSN 0968-0896

Book Section

Castagnolo, Daniele (2012) Chemistry and biological properties of amidinoureas: strategies for the synthesis of unique bioactive hit compounds. In: New Strategies in Chemical Synthesis and Catalysis. Wiley, Weinheim, pp. 97-126. ISBN 978-3527330904